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Table 1 Baseline natural integrase polymorphisms for the HIV-1 clinical isolates used for the in vitro selections with integrase inhibitors

From: Selective resistance profiles emerging in patient-derived clinical isolates with cabotegravir, bictegravir, dolutegravir, and elvitegravir

Isolate ID

GenBank accession number

Subtype

Natural polymorphisms in integrase

14514

KT988124

B

K7R, D10E, S17N, M50I, K111Q, T112V, G123S, T125V, R127K, I220L, Y227F, N232D, D256E

10387

KX7140173

B

D10E, V31I, L45Q, K111E, I113V, G123S, A124T, T125A, R127K, M154I, V201I, D207N, N232D, L234I

10249

KX714014

B

D10E, V31I, L45Q, L101I, K111E, I113V, G123S, A124T, R127K, D207N, N232D, L234I

14624

KX714018

B

D10E, S17N, A23V, L28I, S39C, V72I, L101I, G123S, R127K, N232D

14637

KT988125

B

D10E, E11D, R20K, V31I, S39N, M50I, V72I, S119T, G123S, A124N, R127K, G193E, V201I, D286N

14947

KT988126

B

D10E, E11D, R20K, V31I, S39N, M50I, S119T, G123S, A124N, R127K, G193E, V201I, T218S, D286N

5326

KX714021

B

K7R, D10E, E11D, K14R, V31I, V32I, M50L, V72I, L101I, G123S, A124N, R127K, S195T, I203M, I220L, Y227F, N232D

4742

MG805951

C

D10E, V31I, S39C, V72I, I84M, Q95P, F100Y, L101I, T112V, G123S, A124N, T125A, R127K, D167E, V201I, I203M, K215N, T218L, N232D, L234I, D278A, S283G, R284G

10947

MG805955

C

D6E, D25E, V31I, L45Q, M50I, V72I, P90S, T93S, F100Y, L101I, G106A, T112V, G123S, T125A, R127K, K136Q, V201I, T218I, N232D, L234I, R269K, D278A, S283G, D288N

6343

MG805950

CRF01_AE

D10E, K14R, A21T, V31I, S39N, T112V, G123S, T125A, R127K, G134N, I135V, K136R, D167E, V201I, N232D, L234I, S283G

14515

MG805952

CRF02_AG

D10E, E11D, R20K, A21T, V31I, V72I, L101I, T112V, G123S, T125A, R127K, G134N, K136Q, D167E, V201I, N232D, L234I, V249I, S283G

96USSN20

MG805953

AG

D10E, K14R, V31I, V72I, L101I, T112V, G123S, T125A, R127K, G134N, I135V, K136T, V201I, T206S, N232D, L234I, D256E, R269K, S283G

pNL4.3

 

B

D10E, I113V, S119R, G123S, A124T, R127K, V151I, L234V