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Table 1 Susceptibility of WT and N348 mutant HIV-1 to nevirapine

From: Subunit-specific mutational analysis of residue N348 in HIV-1 reverse transcriptase

Enzyme

IC50 (μM)

Fold Resistance

p66WT/p51WT

0.52 ± 0.04

-

p66N348A/p51N348A

1.77 ± 0.50

3.4

p66N348A/p51WT

0.62 ± 0.07

1.2

p66N348I/p51N348I

4.60 ± 0.45

8.6

p66N348I/p51WT

0.50 ± 0.11

0.97

p66N348L/p51N348L

5.93 ± 0.54

11.4

p66WT/p51N348L

2.96 ± 0.10

5.7

p66N348Q/p51N348Q

1.25 ± 0.13

2.4

p66N348Q/p51WT

0.36 ± 0.05

0.7