Virus strain | Inhibitory activity (Mean ± SD, μM)a | |
---|---|---|
 | IC50 | IC90 |
Laboratory-adapted HIV-1 strains | Â | Â |
   IIIB (X4) | 0.023 ± 0.004 | 0.057 ± 0.004 |
   MN (X4) | 0.151 ± 0.008 | 0.821 ± 0.103 |
   RF (X4R5) | 0.034 ± 0.005 | 0.147 ± 0.059 |
   BaL (R5) | 0.690 ± 0.109 | 2.236 ± 1.184 |
Primary HIV-1 strains | Â | Â |
   UG94103(clade A, X4R5) | 0.561 ± 0.159 | 2.520 ± 1.231 |
   92US657 (clade B, R5) | 2.107 ± 0.263 | 9.357 ± 1.939 |
   93IN101 (clade C, R5) | 1.208 ± 0.535 | 4.946 ± 0.632 |
   BCF02 (clade O, R5) | 0.067 ± 0.004 | 0.188 ± .0.010 |
   Ru570 (clade G, R5) | 4.299 ± 0.298 | 9.332 ± 0.594 |
Drug-resistant HIV-1 | Â | Â |
   AZT-R b | 0.296 ± 0.052 | 1.099 ± 0.773 |
   NL4-3D36Gc | 0.104 ± 0.019 | 0.591 ± 0.059 |
   NL4-3(36G)V38A c | 0.185 ± 0.027 | 0.543 ± 0.026 |
   NL4-3(36G)V38E/N42T c | 0.156 ± 0.082 | 0.992 ± 0.438 |
HIV-2 | Â | Â |
   ROD | 6.079 ± 1.907 | 12.59 ± 3.022 |
SIV | Â | Â |
   mac 251 32H | 0.307 ± 0.174 | 6.128 ± 2.078 |
SHIV | Â | Â |
   SF33A (X4) | 0.189 ± 0.103 | 1.505 ± 0.872 |
   SF162P3 (R5) | 1.312 ± 0.688 | 11.63 ± 5.477 |
HSV | Â | Â |
   HSV-2 strain 333 | 39.06 ± 2.316 | 69.49 ± 3.145 |