Drug | JT-CCR5 Infection | Â | Co-culture JT-CCR5 &explant tissue | Â |
---|---|---|---|---|
 | IC50(μM) | IC90(μM) | IC50(μM) | IC90(μM) |
TDF | 0.04 ± 0.01 | 0.13 ± 0.02 | >10.0 | >10.0 |
IQP-0528 | 0.19 ± 0.07 | 0.43 ± 0.16 | 2.9 ± 0.7 | 10.1 ± 0.7 |
DPV | 0.01 ± 0.01 | 0.03 ± 0.02 | 0.4 ± 0.2 | 1.1 ± 0.3 |
MVC | 1.98 ± 0.85 | 54.5 ± 13.8 | >100 | >100 |
Chol-PIE12 trimer | <0.0001 | 0.009 ± 0.007 | 0.008 ± 0.004 | 0.09 ± 0.01 |
TDF + IQP-0528 | 0.01 ± 0.01 | 0.03 ± 0.02 | 0.5 ± 0.2 | 9.5 ± 0.8 |